PF-299804 (Dacomitinib,PF-00299804)
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC0044 |
Product_name | PF-299804 (Dacomitinib,PF-00299804) |
Category | 抑制剂与激动剂 |
Size | 10mg/50mg/100mg |
Price | 1340.00/2660.00/3880.00 |
Specificity | Target: EGFR. Fields: PF299804 is a potent, irreversible pan-ErbB inhibitor against ErbB1, ErbB2 and ErbB4 with IC50 of 6 nM, 45.7 nM and 73.7 nM, respectively. |
Dilution | IC50: 6 nM (EGFR), 45.7 nM (ERBB2), 73.7 nM (ERBB4)[1] |
Purification | >99% |
Concentration | 靶点:EGFR;IC50: 6 nM (EGFR), 45.7 nM (ERBB2), 73.7 nM (ERBB4)[1] |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | PF299804, Dacomitinib, PF-00299804 |
Molecular Weight | 469.94 |
Notes | PF299804 is a potent, irreversible pan-ErbB inhibitor against ErbB1, ErbB2 and ErbB4 with IC50 of 6 nM, 45.7 nM and 73.7 nM, respectively. |
Instructions | 查看与下载 |
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