PF-299804 (Dacomitinib,PF-00299804)

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0044
Product_name PF-299804 (Dacomitinib,PF-00299804)
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 1340.00/2660.00/3880.00
Specificity Target: EGFR. Fields: PF299804 is a potent, irreversible pan-ErbB inhibitor against ErbB1, ErbB2 and ErbB4 with IC50 of 6 nM, 45.7 nM and 73.7 nM, respectively.
Dilution IC50: 6 nM (EGFR), 45.7 nM (ERBB2), 73.7 nM (ERBB4)[1]
Purification >99%
Concentration 靶点:EGFR;IC50: 6 nM (EGFR), 45.7 nM (ERBB2), 73.7 nM (ERBB4)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername PF299804, Dacomitinib, PF-00299804
Molecular Weight 469.94
Notes PF299804 is a potent, irreversible pan-ErbB inhibitor against ErbB1, ErbB2 and ErbB4 with IC50 of 6 nM, 45.7 nM and 73.7 nM, respectively.
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