VX-680 (MK-0457,Tozasertib)
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC0116 |
Product_name | VX-680 (MK-0457,Tozasertib) |
Category | 抑制剂与激动剂 |
Size | 50mg/100mg |
Price | 660.00/1120.00 |
Specificity | Target: Aurora Kinase. Fields: VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C) |
Dilution | Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C) |
Purification | >98% |
Concentration | 靶点:Aurora Kinase;IC50:Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C) |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | VX680,MK0457,VX 680 (MK 0457,Tozasertib) |
Molecular Weight | 464.59 |
Notes | VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C) |
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