VX-680 (MK-0457,Tozasertib)

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0116
Product_name VX-680 (MK-0457,Tozasertib)
Category 抑制剂与激动剂
Size 50mg/100mg
Price 660.00/1120.00
Specificity Target: Aurora Kinase. Fields: VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
Dilution Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
Purification >98%
Concentration 靶点:Aurora Kinase;IC50:Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername VX680,MK0457,VX 680 (MK 0457,Tozasertib)
Molecular Weight 464.59
Notes VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
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