PHA-739358 (danusertib)

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0140
Product_name PHA-739358 (danusertib)
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 2120.00/6560.00/9440.00
Specificity Target: Aurora Kinase. Fields: Danusertib (PHA-739358) is an Aurora inhibitor for Aurora A/B/C, Bcr-Abl, c-RET and FGFR with IC50 of 13 nM/79 nM/61 nM, 25 nM, 31 nM and 47 nM, respectively.
Dilution IC50: 13 nM (Aurora A), 79 nM (Aurora B), 61 nM (Aurora C)
Purification 99%
Concentration 靶点:Aurora Kinase;IC50: 13 nM (Aurora A), 79 nM (Aurora B), 61 nM (Aurora C)
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
Molecular Weight 474.55
Notes Danusertib (PHA-739358) is an Aurora inhibitor for Aurora A/B/C, Bcr-Abl, c-RET and FGFR with IC50 of 13 nM/79 nM/61 nM, 25 nM, 31 nM and 47 nM, respectively.
Instructions 查看与下载


  • 产品详情
  • 发表文献
  • 用户反馈
  • 相关产品
  • 在线问答