IOX2

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0227
Product_name IOX2
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 1000.00/3880.00/7000.00
Specificity Target: HIF/HIF Prolyl-Hydroxylase. Fields: IOX 2 is a potent inhibitor of HIF-1α prolyl hydroxylase-2 (PHD2) (IC50 = 21 nM). IOX 2 displays over 100-fold selectivity for PHD2 over factor inhibiting HIF-1 (FIH-1) and histone demethylases.
Dilution IC50: 22 nM (PHD2)[1]
Purification >98%
Concentration 靶点:HIF/HIF Prolyl-Hydroxylase;IC50: 22 nM (PHD2)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername IOX-2; IOX2; IOX 2
Molecular Weight 352.34
Notes IOX 2 is a potent inhibitor of HIF-1α prolyl hydroxylase-2 (PHD2) (IC50 = 21 nM). IOX 2 displays over 100-fold selectivity for PHD2 over factor inhibiting HIF-1 (FIH-1) and histone demethylases.
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