| Catalog_no |
ADMC0675 |
| Product_name |
GSK923295 |
| Category |
抑制剂与激动剂 |
| Size |
10mg/50mg/100mg |
| Price |
2000.00/7000.00/12220.00 |
| Specificity |
Target: Kinesin . Fields: GSK923295 is a first-in-class, specific allosteric inhibitor of CENP-E kinesin motor ATPase with Ki of 3.2 nM, and less potent to mutant I182 and T183. Phase 1. Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Dilution |
Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Purification |
>98% |
| Concentration |
靶点：Kinesin;IC50：Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Storage_stability |
2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
| othername |
GSK-923295 |
| Molecular Weight |
592.13 |
| Notes |
GSK923295 is a first-in-class, specific allosteric inhibitor of CENP-E kinesin motor ATPase with Ki of 3.2 nM, and less potent to mutant I182 and T183. Phase 1. Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Instructions |
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