Brexpiprazole(OPC34712)

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0865
Product_name Brexpiprazole(OPC34712)
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 780.00/1220.00/1880.00
Specificity Target: 5-HT Receptor . Fields: Brexpiprazole is a novel D2 dopamine partial agonist. Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1]
Dilution Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1]
Purification >98%
Concentration 靶点:5-HT Receptor;IC50:Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername OPC 34712; OPC34712; OPC-34712
Molecular Weight 433.57
Notes Brexpiprazole is a novel D2 dopamine partial agonist. Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1]
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