Brexpiprazole(OPC34712)
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC0865 |
Product_name | Brexpiprazole(OPC34712) |
Category | 抑制剂与激动剂 |
Size | 10mg/50mg/100mg |
Price | 780.00/1220.00/1880.00 |
Specificity | Target: 5-HT Receptor . Fields: Brexpiprazole is a novel D2 dopamine partial agonist. Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1] |
Dilution | Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1] |
Purification | >98% |
Concentration | 靶点:5-HT Receptor;IC50:Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1] |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | OPC 34712; OPC34712; OPC-34712 |
Molecular Weight | 433.57 |
Notes | Brexpiprazole is a novel D2 dopamine partial agonist. Ki: 0.12 nM (5-HT1A), 0.3 nM (D2L), 0.47 nM (5-HT2A)[1] |
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