RVX-208

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0888
Product_name RVX-208
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 1120.00/3880.00/7000.00
Specificity Target: Epigenetic Reader Domain . Fields: RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist. IC50: 510±41 nM (BD2), 87±10 μM (BD1)
Dilution IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
Purification >98%
Concentration 靶点:Epigenetic Reader Domain;IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername Apabetalone; RVX-000222; RVX208; RVX 208; RVX000222; RVX 000222
Molecular Weight 370.4
Notes RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist. IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
Instructions 查看与下载


  • 产品详情
  • 发表文献
  • 用户反馈
  • 相关产品
  • 在线问答