JNJ-42041935

日期:2018-09-05 17:14 人气:
Catalog_no ADMC0986
Product_name JNJ-42041935
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 2120.00/8440.00/15200.00
Specificity Target: HIF/HIF Prolyl-Hydroxylase. Fields: JNJ-42041935 is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes. pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1]
Dilution pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1]
Purification >98%
Concentration 靶点:HIF/HIF Prolyl-Hydroxylase;IC50:pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername JNJ 42041935,JNJ42041935,HIF-PHD Inhibitor II
Molecular Weight 346.65
Notes JNJ-42041935 is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes. pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1]
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