JNJ-42041935
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC0986 |
Product_name | JNJ-42041935 |
Category | 抑制剂与激动剂 |
Size | 10mg/50mg/100mg |
Price | 2120.00/8440.00/15200.00 |
Specificity | Target: HIF/HIF Prolyl-Hydroxylase. Fields: JNJ-42041935 is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes. pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1] |
Dilution | pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1] |
Purification | >98% |
Concentration | 靶点:HIF/HIF Prolyl-Hydroxylase;IC50:pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1] |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | JNJ 42041935,JNJ42041935,HIF-PHD Inhibitor II |
Molecular Weight | 346.65 |
Notes | JNJ-42041935 is a potent (pKi = 7.3-7.9), 2-oxoglutarate competitive, reversible, and selective inhibitor of PHD enzymes. pKi: 7.91±0.04 (PHD1), 7.29 ±0.05 (PHD2), 7.65±0.09(PHD3)[1] |
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