Nazartinib(EGF816)

日期:2018-09-05 17:14 人气:
Catalog_no ADMC1216
Product_name Nazartinib(EGF816)
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 5560.00/16660.00/23340.00
Specificity Target: EGFR. Fields: Nazartinib(EGF816) is a novel covalent inhibitor of mutant-selective EGFR; overcomes T790M-mediated resistance in NSCLC. Ki: 31 nM (EGFR(L858R/790M) mutant)[2]
Dilution Ki: 31 nM (EGFR(L858R/790M) mutant)[2]
Purification >98%
Concentration 靶点:EGFR;IC50:Ki: 31 nM (EGFR(L858R/790M) mutant)[2]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername EGF-816,EGF 816
Molecular Weight 495.02
Notes Nazartinib(EGF816) is a novel covalent inhibitor of mutant-selective EGFR; overcomes T790M-mediated resistance in NSCLC. Ki: 31 nM (EGFR(L858R/790M) mutant)[2]
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