IPI-549

日期:2018-09-05 17:14 人气:
Catalog_no ADMC1236
Product_name IPI-549
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 1660.00/3880.00/7000.00
Specificity Target: PI3K. Fields: IPI-549 is an orally administered immuno-oncology development candidate that selectively inhibits PI3K-gamma. IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1]
Dilution IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1]
Purification >98%
Concentration 靶点:PI3K;IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername IPI549,IPI 549
Molecular Weight 528.2
Notes IPI-549 is an orally administered immuno-oncology development candidate that selectively inhibits PI3K-gamma. IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1]
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