IPI-549
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC1236 |
Product_name | IPI-549 |
Category | 抑制剂与激动剂 |
Size | 10mg/50mg/100mg |
Price | 1660.00/3880.00/7000.00 |
Specificity | Target: PI3K. Fields: IPI-549 is an orally administered immuno-oncology development candidate that selectively inhibits PI3K-gamma. IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1] |
Dilution | IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1] |
Purification | >98% |
Concentration | 靶点:PI3K;IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1] |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | IPI549,IPI 549 |
Molecular Weight | 528.2 |
Notes | IPI-549 is an orally administered immuno-oncology development candidate that selectively inhibits PI3K-gamma. IC50: 16 nM (PI3Kγ), 3.2 μM (PI3Kα), 3.5 μM (PI3Kβ), >8.4 μM (PI3Kδ)[1] |
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