(±)-SLV319

日期:2018-09-05 17:14 人气:
Catalog_no ADMC1362
Product_name (±)-SLV319
Category 抑制剂与激动剂
Size 10mg/50mg/100mg
Price 1780.00/7340.00/12780.00
Specificity Target: Cannabinoid Receptor. Fields: (±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
Dilution IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
Purification >98%
Concentration 靶点:Cannabinoid Receptor;IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
Storage_stability 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othername SLV 319,SLV-319
Molecular Weight 487.4
Notes (±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
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