(±)-SLV319
日期:2018-09-05 17:14 人气:
Catalog_no | ADMC1362 |
Product_name | (±)-SLV319 |
Category | 抑制剂与激动剂 |
Size | 10mg/50mg/100mg |
Price | 1780.00/7340.00/12780.00 |
Specificity | Target: Cannabinoid Receptor. Fields: (±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2] |
Dilution | IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2] |
Purification | >98% |
Concentration | 靶点:Cannabinoid Receptor;IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2] |
Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
othername | SLV 319,SLV-319 |
Molecular Weight | 487.4 |
Notes | (±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2] |
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