抑制剂与激动剂

Catalog_noADMC0052
Product_nameI-BET151 (GSK1210151A)
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1340.00/4000.00/7000.00
SpecificityTarget: Epigenetic Reader Domain. Fields: I-BET151 (GSK1210151A) is a novel selective BET inhibitor for BRD2, BRD3 and BRD4 with IC50 of 0.5 μM, 0.25 μM, and 0.79 μM, respectively.
DilutionpIC50: 6.1 (BRD4), 6.3 (BRD2), 6.6 (BRD3)[1]
Purification>98%
Concentration靶点:Epigenetic Reader Domain;IC50:p 6.1 (BRD4), 6.3 (BRD2), 6.6 (BRD3)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameGSK-1210151A,IBET151,I-BET-151,I BET 151,IBET-151,IBET 151,GSK 1210151A
Observed_band415.44
NotesI-BET151 (GSK1210151A) is a novel selective BET inhibitor for BRD2, BRD3 and BRD4 with IC50 of 0.5 μM, 0.25 μM, and 0.79 μM, respectively.
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