抑制剂与激动剂

Catalog_noADMC0095
Product_nameBIX02188 (BIX 02188)
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price2840.00/8620.00/15520.00
SpecificityTarget: MEK. Fields: BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
Dilution
Purification>98%
Concentration靶点:MEK;IC50:No data
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameBIX 02188; BIX02188; BIX-02188
Observed_band426.51
NotesBIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
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