抑制剂与激动剂

Catalog_noADMC0116
Product_nameVX-680 (MK-0457,Tozasertib)
Category抑制剂与激动剂
Size50mg/100mg
Price660.00/1120.00
SpecificityTarget: Aurora Kinase. Fields: VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
DilutionKi: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
Purification>98%
Concentration靶点:Aurora Kinase;IC50:Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameVX680,MK0457,VX 680 (MK 0457,Tozasertib)
Observed_band464.59
NotesVX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively. Ki: 0.6 nM (Aurora A), 18 nM (Aurora B), 4.6 nM (Aurora C)
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