抑制剂与激动剂

Catalog_noADMC0221
Product_nameLY2835219(Abemaciclib)
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1000.00/2120.00/2660.00
SpecificityTargetTargets the CDK4 (cyclin D1) and CDK6 (cyclin D3) cell cycle pathway, with potential antineoplastic activity. IC50: 2 nM (CDK4), 10 nM (CDK6)
DilutionIC50: 2 nM (CDK4), 10 nM (CDK6)
Purification>99%
Concentration靶点:CDK;IC50: 2 nM (CDK4), 10 nM (CDK6)
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameLY2835219; LY-2835219; LY 2835219
Observed_band602.7
NotesLY2835219 is an orally available cyclin-dependent kinase (CDK) inhibitor that targets the CDK4 (cyclin D1) and CDK6 (cyclin D3) cell cycle pathway, with potential antineoplastic activity. IC50: 2 nM (CDK4), 10 nM (CDK6)
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