抑制剂与激动剂

Catalog_noADMC0321
Product_nameBI-D1870
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price2340.00/6060.00/10900.00
SpecificityTarget: Ribosomal S6 Kinase (RSK). Fields: BI-D1870 is a small molecule, specific inhibitor of p90 RSK (ribosomal S6 kinase) isoforms RSK1, RSK2, RSK3 and RSK4, both in vitro and in vivo, with IC50s are 31 nM, 24 nM, 18 nM, 15 nM, respectively.
Dilution
Purification>98%
Concentration靶点:Ribosomal S6 Kinase (RSK);IC50:No data
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameBID1870
Observed_band391.42
NotesBI-D1870 is a small molecule, specific inhibitor of p90 RSK (ribosomal S6 kinase) isoforms RSK1, RSK2, RSK3 and RSK4, both in vitro and in vivo, with IC50s are 31 nM, 24 nM, 18 nM, 15 nM, respectively.
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