抑制剂与激动剂

Catalog_noADMC0348
Product_nameGSK-1070916
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1660.00/4440.00/7780.00
SpecificityTarget: Aurora Kinase. Fields: GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B/C with IC50 of 3.5 nM/6.5 nM; displays >100-fold selectivity against the closely related Aurora A-TPX2 complex(IC50=490 nM).
Dilution
Purification>98%
Concentration靶点:Aurora Kinase;IC50:No data
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameGSK1070916; GSK 1070916
Observed_band507.63
NotesGSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B/C with IC50 of 3.5 nM/6.5 nM; displays >100-fold selectivity against the closely related Aurora A-TPX2 complex(IC50=490 nM).
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