| Catalog_no | ADMC0349 |
| Product_name | Omipalisib(GSK-458) |
| Category | 抑制剂与激动剂 |
| Size | 10mg/50mg/100mg |
| Price | 1780.00/4660.00/8400.00 |
| Specificity | Target: PI3K. Fields: GSK2126458 is a highly selective and potent inhibitor of PI3K with Ki of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2 , respectively. Ki: 0.019 nM (p110α), 0.13 nM (p110β), 0.024 nM (p110δ), 0. |
| Dilution | Ki: 0.019 nM (p110α), 0.13 nM (p110β), 0.024 nM (p110δ), 0.06 nM (p110γ), 0.18 nM (mTORC1), 0.3 nM (mTORC2) |
| Purification | >98% |
| Concentration | 靶点：PI3K;IC50：Ki: 0.019 nM (p110α), 0.13 nM (p110β), 0.024 nM (p110δ), 0.06 nM (p110γ), 0.18 nM (mTORC1), 0.3 nM (mTORC2) |
| Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
| othername | GSK212; GSK-2126458; GSK 2126458; GSK-212; GSK 212，GSK458，GSK 458,GSK2126458 |
| Observed_band | 505.5 |
| Notes | GSK2126458 is a highly selective and potent inhibitor of PI3K with Ki of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2 , respectively. Ki: 0.019 nM (p110α), 0.13 nM (p110β), 0.024 nM (p110δ), 0.06 nM (p110γ), 0.18 nM |
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