抑制剂与激动剂

Catalog_noADMC0508
Product_nameRibociclib (LEE011)
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price880.00/1340.00/2000.00
SpecificityTargetTargeting cyclin D1/CDK4 and cyclin D3/CDK6 cell cycle pathway, with potential antineoplastic activity. IC50: 10/39 nM (CDK4/6)[1]
DilutionIC50: 10/39 nM (CDK4/6)[1]
Purification>99%
Concentration靶点:CDK;IC50: 10/39 nM (CDK4/6)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameLEE 011; LEE-011,Ribociclib,LEE011
Observed_band434.54
NotesLEE011 is an orally available cyclin-dependent kinase (CDK) inhibitor targeting cyclin D1/CDK4 and cyclin D3/CDK6 cell cycle pathway, with potential antineoplastic activity. IC50: 10/39 nM (CDK4/6)[1]
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