400-921-8278
| Catalog_no | ADMC0523 |
| Product_name | Torkinib (PP242) |
| Category | 抑制剂与激动剂 |
| Size | 10mg/50mg/100mg |
| Price | 820.00/1960.00/3520.00 |
| Specificity | TargetTargets both mTOR complexes with >10- and 100-fold selectivity for mTOR than PI3Kδ or PI3Kα/β/γ, respectively; also showed slightly weaker activity against BRD4 (Kd= 1.7 uM). |
| Dilution | IC50: 8 nM (mTOR), 100 nM (p110δ), 410 nM (DNA-PK), 410 nM (PDGFR)[1] |
| Purification | >98% |
| Concentration | 靶点：mTOR;IC50： 8 nM (mTOR), 100 nM (p110δ), 410 nM (DNA-PK), 410 nM (PDGFR)[1] |
| Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
| othername | TORKinib,PP242; PP-242,PP 242 |
| Observed_band | 308.34 |
| Notes | PP242 is a selective mTOR inhibitor with IC50 of 8 nM; targets both mTOR complexes with >10- and 100-fold selectivity for mTOR than PI3Kδ or PI3Kα/β/γ, respectively; also showed slightly weaker activity against BRD4 (Kd= 1.7 uM). |
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