抑制剂与激动剂

Catalog_noADMC0611
Product_nameIBMX(NSC165960; SC2964)
Category抑制剂与激动剂
Size50mg/100mg
Price560.00/1000.00
SpecificityTarget: Phosphodiesterase (PDE) . Fields: IBMX(NSC165960; SC2964) is a competitive nonselective PDEs inhibitor with IC50 of 2-50 uM but does not inhibit PDE8 or PDE9; nonselective adenosine receptor antagonist.
DilutionIC50: 6.5±1.2 μM(PDE3), 26.3±3.9 μM (PDE4), 31.7±5.3 μM (PDE5)[1]
Purification>98%
Concentration靶点:Phosphodiesterase (PDE);IC50: 6.5±1.2 μM(PDE3), 26.3±3.9 μM (PDE4), 31.7±5.3 μM (PDE5)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameIMX; Isobutylmethylxanthine; Methylisobutylxanthine; NSC165960; SC2964
Observed_band222.24
NotesIBMX(NSC165960; SC2964) is a competitive nonselective PDEs inhibitor with IC50 of 2-50 uM but does not inhibit PDE8 or PDE9; nonselective adenosine receptor antagonist.
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