| Catalog_no | ADMC0675 |
| Product_name | GSK923295 |
| Category | 抑制剂与激动剂 |
| Size | 10mg/50mg/100mg |
| Price | 2000.00/7000.00/12220.00 |
| Specificity | Target: Kinesin . Fields: GSK923295 is a first-in-class, specific allosteric inhibitor of CENP-E kinesin motor ATPase with Ki of 3.2 nM, and less potent to mutant I182 and T183. Phase 1. Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Dilution | Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Purification | >98% |
| Concentration | 靶点：Kinesin;IC50：Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
| Storage_stability | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
| othername | GSK-923295 |
| Observed_band | 592.13 |
| Notes | GSK923295 is a first-in-class, specific allosteric inhibitor of CENP-E kinesin motor ATPase with Ki of 3.2 nM, and less potent to mutant I182 and T183. Phase 1. Ki: 3.2 nM (human CENP-E), 1.6 nM (canine CENP-E)[1] |
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