抑制剂与激动剂

Catalog_noADMC0888
Product_nameRVX-208
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1120.00/3880.00/7000.00
SpecificityTarget: Epigenetic Reader Domain . Fields: RVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist. IC50: 510±41 nM (BD2), 87±10 μM (BD1)
DilutionIC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
Purification>98%
Concentration靶点:Epigenetic Reader Domain;IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameApabetalone; RVX-000222; RVX208; RVX 208; RVX000222; RVX 000222
Observed_band370.4
NotesRVX-208(RVX 000222) is a small molecule that increases apolipoprotein A-I and high-density lipoprotein cholesterol in vitro and in vivo; is a BET bromodomain antagonist. IC50: 510±41 nM (BD2), 87±10 μM (BD1)[1]
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