抑制剂与激动剂

Catalog_noADMC0948
Product_namePalbociclib isethionate
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price780.00/1000.00/1440.00
SpecificityTarget: CDK . Fields: Palbociclib isethionate(PD-0332991 isethionate) is a highly specific inhibitor of Cdk4 (IC50=11 nM) and Cdk6 (IC50=16 nM), having no activity against a panel of 36 additional protein kinases.
DilutionIC50: 11 nM (CDK4), 16 nM (CDK6)
Purification>98%
Concentration靶点:CDK;IC50: 11 nM (CDK4), 16 nM (CDK6)
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernamePD0332991; PD-0332991; PD 0332991
Observed_band573.66
NotesPalbociclib isethionate(PD-0332991 isethionate) is a highly specific inhibitor of Cdk4 (IC50=11 nM) and Cdk6 (IC50=16 nM), having no activity against a panel of 36 additional protein kinases.
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