抑制剂与激动剂

Catalog_noADMC1355
Product_nameUK-371804
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price2340.00/7220.00/10560.00
SpecificityTarget: Ser/Thr Protease. Fields: UK-371804 is a potent and selective uPA inhibitor with excellent enzyme potency (Ki 10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). Ki: 10 nM (uPA)[1]
DilutionKi: 10 nM (uPA)[1]
Purification>98%
Concentration靶点:Ser/Thr Protease;IC50:Ki: 10 nM (uPA)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameUK371804,UK 371804
Observed_band385.06
NotesUK-371804 is a potent and selective uPA inhibitor with excellent enzyme potency (Ki 10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). Ki: 10 nM (uPA)[1]
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