抑制剂与激动剂

Catalog_noADMC1362
Product_name(±)-SLV319
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1780.00/7340.00/12780.00
SpecificityTarget: Cannabinoid Receptor. Fields: (±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
DilutionIC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
Purification>98%
Concentration靶点:Cannabinoid Receptor;IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameSLV 319,SLV-319
Observed_band487.4
Notes(±)-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. IC50: 22 nM (CB-1)[1]; Ki: 7.8 nM (CB-1)[2]
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